Publication
Number of items: 15.
None
NK1 antagonists based on seven membered lactam scaffolds. (2006)
J. M. Elliott,
E. J. Carlson,
G. G. Chcchi,
O. Dirat,
M. Dominguez,
U. Gerhard,
R. Jelley,
A. B. Jones,
M. M. Kurtz,
K. I. Tsao
and
A. Wheeldon
Conformationally restricted indolopiperidine derivatives as potent CCR2B receptor antagonists. (2001)
Jason Witherington,
Vincent Bordas,
Dave G. Cooper,
Ian T. Forbes,
Andrew D. Gribble,
Robert J. Ife,
Theo Berkhout,
Jayneeta Gohil
and
Pieter H. E. Groot
CCR2B receptor antagonists : Conversion of a weak HTS hit to a potent lead compound. (2000)
Ian T. Forbes,
David G. Cooper,
Emma K. Dodds,
Deirdre M. B. Hickey,
Robert J. Ife,
Malcolm Meeson,
Martin Stockley,
Theo Berkhout,
Jayneeta Gohil,
Pieter H. E. Groot
and
Kitty E. Moores
Synthesis of conformationally constrained analogues of BRL32872 : Determination of stereochemistry and related pharmacological properties. (1997)
M. Souchet,
M.-C. Forest,
B. Cheval,
S. Rouanet,
J.-F. Faivre,
A. Bril,
U. Gerhard
and
R.J. Smith
Aryl sulfones : A new class of γ-secretase inhibitors. (2005)
M. Teall,
P. Oakley,
T. Harrison,
D. Shaw,
E. Kay,
J. Elliott,
U. Gerhard,
J.L. Castro,
M. Shearman,
R.G. Ball
and
N.N. Tsou
The free energy change of restricting a bond rotation in the binding of peptide analogues to vancomycin group antibiotics. (1993)
U. Gerhard,
M.S. Searle
and
D.H. Williams
Investigation of the protein alkylation sites of the STAT3:STAT3 inhibitor Stattic by mass spectrometry. (2013)
Sibylle Heidelberger,
Giovanna Zinzalla,
Dyeison Antonow,
Samantha Essex,
B. Piku Basu,
Jonathan Palmer,
Jarmila Husby,
Paul J. M. Jackson,
Khondaker M. Rahman,
Andrew F. Wilderspin,
Mire Zloh
and
David E. Thurston
Inhibitors of multidrug resistance (MDR) have affinity for MDR substrates. (2004)
Mire Zloh,
G.W. Kaatz
and
S. Gibbons
Target fishing and docking studies of the novel derivatives of aryl-aminopyridines with potential anticancer activity. (2012)
S. Erić,
J. Antić Stanković,
V. Savić,
S. Ke,
T. Barata,
T. Solmajer,
Z. Juranić
and
Mire Zloh
Sequences in the HSP90 promoter form G-quadruplex structures with selectivity for disubstituted phenyl bis-oxazole derivatives. (2012)
Stephan A. Ohnmacht,
Marialuisa Micco,
Vanessa Petrucci,
Alan K. Todd,
Anthony P. Reszka,
Mekala Gunaratnam,
Marta A. Carvalho,
Mire Zloh
and
Stephen Neidle
2-Hexadecynoic acid inhibits plasmodial FAS-II enzymes and arrests erythrocytic and liver stage Plasmodium infections. (2010)
Deniz Tasdemir,
David Sanabria,
Ina L Lauinger,
Alice Tarun,
Rob Herman,
Remo Perozzo,
Mire Zloh,
Stefan H. Kappe,
Reto Brun
and
Néstor M Carballeira
An analysis of the 'legal high' mephedrone. (2010)
Simon Gibbons
and
Mire Zloh
Public
Discovery of inhibitors of the pentein superfamily protein dimethylarginine dimethylaminohydrolase (DDAH), by virtual screening and hit analysis. (2007)
B. Hartzoulakis,
S. Rossiter,
H. Gill,
E. Steinke,
P.J. Gane,
R. Hurtado-Guerrero,
J.M. Leiper,
P. Vallance,
J. Murray-Rust
and
D.L. Selwood
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Halogenated indole-3-acetic acids as oxidatively activated prodrugs with potential for targeted cancer therapy. (2002)
S. Rossiter,
L.K. Folkes
and
P. Wardman
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Synthesis and anthelmintic properties of arylquinolines with activity against drug resistant nematodes. (2005)
S. Rossiter,
J. M. Peron,
P.J. Whitfield
and
K. Jones
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